Opioid Antagonism in Humans: A Primer on Optimal Dose and Timing for Central Mu-Opioid Receptor Blockade
Martin Trøstheim, Marie Eikemo, Jan Haaker, J. James Frost, Siri Leknes
The paper analyzes opioid receptor blockade using PET data and models to determine optimal doses and timing for naloxone and naltrexone in humans.
Neuropsychopharmacology · Aug 17, 2022Peer-reviewedNeuroscience