Predicting PROTAC-targeted Degradation and Designing Androgen Receptor Degraders with AiPROTAC
Li Zhang, Renhong Sun, Xia Li, Chaowei Ren, Yahui Long, Wenjuan Tan, Xiaolong Wang, Ke Zou, Xiaobao Yang, Min Wu, Xiaoli Li, Xing Chen
AiPROTAC predicts PROTAC degradation potential and designs an androgen receptor degrader, outperforming existing models and showing improved in vitro efficacy.
bioRxiv · Feb 26, 2025 · PreprintBioinformatics