Discovery of molecular glues that bind FKBP12 and novel targets using DNA-barcoded libraries
Trevor A. Zandi, M.J. Romanowski, Jessica S. Viscomi, Karl Gunderson, Zher Yin Tan, Bingqi Tong, Simone Bonazzi, Frédéric J. Zécri, Stuart L. Schreiber, Gregory A. Michaud
This study identifies novel FKBP12 molecular glues and their targets using DNA-encoded libraries, showing FKBP12-dependent recruitment to BRD9 and QDPR.
Nature Communications · Apr 22, 2026Peer-reviewedBiophysics