Di-berberine conjugates as chemical probes of Pseudomonas aeruginosa MexXY-OprM efflux function and inhibition
L. G. Kavanaugh, A. R. Mahoney, D. Dey, W. M. Wuest, G. L. Conn
This study optimizes berberine derivatives to create di-berberine conjugates that enhance aminoglycoside efficacy by inhibiting Pseudomonas aeruginosa MexY efflux pump function.
bioRxiv · Mar 24, 2023 · PreprintMicrobiology