Cancer BiologybioRxivPreprint
Mirror-image mRNA display uncovers isoform-selective D-peptide macrocycles targeting a cryptic KRAS pocket
Matthew J. Mitcheltree, Nicole Boo, Nicolas C. Boyer…·Kaustav Biswas
This paper uses mirror-image mRNA display to discover D-peptide macrocycles targeting a new KRAS binding site, showing selectivity and efficacy in inhibiting KRAS-mutant cells.
DOI 10.64898/2026.05.20.726527