mPD5, a peripherally restricted PICK1 inhibitor for treating chronic pain
K. L. Jensen, N. R. Christensen, C. M. Goddard, S. E. Jager, I. B. Kanneworff, A. Jakobsen, G. Noes-Holt, L. Jimenez-Fernandez, E. G. Peck, L. Sivertsen, R. C. Baro, G. A. Houser, F. P. Mayer, M. D. del Castillo, M. L. Topp, , K. L. Madsen
This paper develops mPD5, a peripherally restricted PICK1 inhibitor that reduces chronic pain and associated symptoms in mice without significant side effects.
bioRxiv · Mar 3, 2023 · PreprintPharmacology & Toxicology