Three nitrogen atoms turn old kinase inhibitors into new targetable remedy
Balázs Besztercei, Réka Antal, Leena Tähtivaara, Birgitta Lappeteläinen, Niina Jääskeläinen, Attila Szappanos, Ákos Lukáts, Alexandra Pal-Kajtar, András Budai, András Dénes Marton, Marcell Stifter-Mursits, László Hiripi, György Tibor Balogh, Marc Cerrada‐Gimenez, Krisztián A. Kovács
This paper introduces photoactivatable VEGFR2 inhibitors that enhance retinal disease treatment by light-triggered activation, reducing required doses and systemic exposure.
Journal of Medicinal Chemistry · Oct 4, 2026Peer-reviewedPharmacology & Toxicology