Identification of actionable targeted protein degradation effector sites through Site-specific Ligand Incorporation-induced Proximity (SLIP)
Zhangping Xiao, Efthymios-Spyridon Gavriil, Fangyuan Cao, Xinyue Zhang, Stan Xiaogang Li, Sergei Kotelnikov, Patrycja Michalska, Friederike Marte, Chloe Huang, Yudi Lu, Yunxuan Zhang, Erika Bernardini, Dima Kozakov, Edward W. Tate
The paper introduces a chemical-genetic platform called SLIP to identify actionable sites on effector proteins for targeted protein degradation.
Journal of the American Chemical Society · Jun 10, 2025Peer-reviewedMolecular Biology