Head-to-tail peptide cyclization: new directions and application to urotensin II and Nrf2
Yasaman Karami, Samuel Murail, Julien Giribaldi, Benjamin Lefranc, Florian Defontaine, Olivier Lesouhaitier, Jérôme Leprince, Sjoerd J. de Vries, Pierre Tufféry
The paper introduces a framework for rational head-to-tail peptide cyclization using protein structure data, demonstrating improved conformation prediction and successful application to Nrf2 and urotensin II peptides.
bioRxiv · Jan 5, 2022 · PreprintBioinformatics