Localized in vivo prodrug activation using radionuclides
Jeremy M. Quintana, Fangchao Jiang, Mikyung Kang, Víctor Valladolid Onecha, Arda Könik, Lei Qin, Victoria E. Rodriguez, Huiyu Hu, Nicholas Borges, Ishaan Khurana, Leou Ismael Banla, Mariane Le Fur, Peter D. Caravan, Jan Schuemann, Alejandro Bertolet, , Thomas S.C. Ng
This paper demonstrates RAiDER, a method using radionuclides to locally activate prodrugs at tumor sites, showing significant cytotoxicity enhancement and reduced off-target effects.
Journal of Nuclear Medicine · Jan 1, 2025Peer-reviewedBioengineering