Click-to-Release: Cleavable Radioimmunoimaging with 89Zr-DFO-Trans-Cyclooctene-Trastuzumab Increases Tumor-to-Blood Ratio
M. Vlastara, R. Rossin, F. J. Hoeben, K. E. de Roode, M. Boswinkel, L. H. Kleijn, J. Nagarajah, M. Rijpkema, M. S. Robillard
This paper demonstrates a click-to-release method to improve PET imaging by reducing background signals through selective cleavage of radiolabeled antibodies in mice.
bioRxiv · Mar 27, 2023 · PreprintPharmacology & Toxicology