Illuminating kinase inhibitors biology by cell signaling profiling.
A. Medvedev, S. Makarov, L. A. Medvedeva, E. Martsen, K. L. Gorman, B. Lin, S. S. Makarov
This paper introduces a method to evaluate kinase inhibitors by profiling transcription factor activity, revealing consensus signatures that indicate on-target biological effects.
bioRxiv · Apr 3, 2022 · PreprintPharmacology & Toxicology