Paired activity learning supports systematic identification of mutant-selective EGFR inhibitors
Jie Zhu, Weikaixin Kong, Liting Huang, Zejia Z Song, Huiyan Ying, Kari J. Kurppa, Mitro Miihkinen, Sujie Zhu, Tero A. Aittokallio
The paper develops a computational-experimental framework to identify mutant-selective EGFR inhibitors by leveraging paired activity measurements and structural analysis.
bioRxiv · Oct 26, 2026 · PreprintBioinformatics