Pharmacological characterization of seven human histamine H3 receptor isoforms
M. Gao, M. E. Dekker, R. Leurs, H. F. Vischer
This study pharmacologically characterizes seven human H3R isoforms, finding differences in agonist and inverse agonist binding affinities, with implications for drug discovery.
bioRxiv · Dec 6, 2023 · PreprintPharmacology & Toxicology