BiochemistryJournal of Medicinal ChemistryPeer-reviewed
Discovery of the First-in-class G9a/GLP PROTAC Degrader
Julia Velez, Yulin Han, Hyerin Yim…·Jian Jun Jin
This paper discovers a first-in-class PROTAC degrader for G9a/GLP, showing effective degradation and superior anticancer activity compared to existing inhibitors.