BiochemistryeLifePeer-reviewed
Kinases in motion: impact of protein and small molecule interactions on kinase conformations
Valentina Kugler, Selina Schwaighofer, Andreas Feichtner…·Eduard Stefan
This study uses KinCon-reporter technology to analyze conformational changes in disease-associated kinases upon drug, regulatory protein, and pathway activation interactions, revealing insights into therapeutic strategies.
6 citations