The ion channel TRPM8 is a direct target of the immunosuppressant rapamycin in primary sensory neurons
José Miguel Arcas, Khalid Oudaha, Alejandro González, Jorge Fernández‐Trillo, Francisco Andrés Peralta, Júlia Castro‐Marsal, Seyma Poyraz, Francisco José Taberner, Salvador Sala, Elvira de la Peña, Ana Gomis, Félix Viana
This study identifies TRPM8 ion channels as direct targets of rapamycin in sensory neurons, showing RAP activates TRPM8 and induces tearing via TRPM8-dependent mechanisms.
British Journal of Pharmacology · May 13, 2024Peer-reviewedNeuroscience