Cancer BiologybioRxiv
Dual mechanism estrogen receptor inhibitors
J. Min, J. C. Nwachukwu, S. Srinivasan…·K. W. Nettles
This paper develops dual-mechanism ER inhibitors that use two distinct targeting moieties to suppress ER activity in breast cancer cells and resistance models.
DOI 10.1073/pnas.2101657118