Pharmacology & ToxicologyJournal of Medicinal ChemistryPeer-reviewed
Discovery of the first-efficacious A2AR negative allosteric modulators for high adenosine cancer immunotherapies
Margot Boujut, Margaux Héritier, Aurélie Gouiller…·Léonardo Scapozza
The paper identifies potent A2AR negative allosteric modulators through high-throughput screening and SAR analysis, showing their efficacy in high-adenosine conditions for safer cancer immunotherapies.
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