Novel naphthyridones targeting Pannexin 1 for colitis management
Wen‐Yun Hsueh, Yiling Wu, Meng‐Tzu Weng, Shin‐Yun Liu, Jascinta P. Santavanond, Yi‐Chung Liu, Ching‐I Lin, Cheng‐Nong Lai, Yi‐Ru Lu, Jing Yin Hsu, Hong‐Yu Gao, Jinq‐Chyi Lee, Shu‐Chen Wei, Pingchiang C. Lyu, Ivan K. H. Poon, , Yu‐Hsin Chiu
The paper identifies a novel naphthyridone inhibitor of PANX1 with reduced off-target effects, showing efficacy in a mouse model of IBD.
Advanced Science · Dec 30, 2024Peer-reviewedMolecular Biology