BioinformaticsACS OmegaPeer-reviewed
A deep learning approach for the discovery of tumor-targeting small organic ligands from DNA-Encoded Chemical Libraries
Wen Torng, Ilaria Biancofiore, Sebastian Oehler…·Jianwen A. Feng
The paper uses deep learning to identify tumor-targeting ligands from DNA-encoded chemical libraries against CAIX, finding 70% of novel hits show submicromolar activity.