Structural basis of saccharine derivative inhibition of carbonic anhydrase IX
Jānis Leitāns, Andris Kazāks, Jānis Bogans, Claudiu Trandafir Supuran, Ināra Akopjana, Jekaterīna Ivanova, Raivis Žalubovskis, Kaspars Tārs
This study investigates the binding of saccharine derivatives to hCA IX using crystallography, revealing structural insights for designing selective inhibitors.
bioRxiv · Nov 1, 2023 · PreprintMolecular Biology