A broad set of synthetic cannabinoid receptor agonists inhibit the cardiac voltage-gated potassium channel hERG
Nina E. Ottosson, Damon J.A. Frampton, Tanadet Pipatpolkai, Caitlyn Norman, Urban Karlsson, Amaia Jauregi‐Miguel, Maryke Venter, Akshay Sridhar, Hans Peter Larsson, Henrik Gréen, Sara I. Liin
This study investigates how synthetic cannabinoid receptor agonists affect cardiac ion channels, finding that most inhibit hERG and some also inhibit KV7.1/KCNE1.
Acta Pharmacologica Sinica · Jul 21, 2026Peer-reviewedPharmacology & Toxicology