BiochemistryACS Chemical BiologyPeer-reviewed
Overcoming Ligand Discovery Challenges: Developing Peptide-Based Tracers for SPSB2
Christopher Lenz, Lewis Elson, Johannes Dopfer…·Stefan Knapp
This study develops peptide-based tracers for SPSB2 E3 ligase by conjugating cell-penetrating peptides to degrons, enabling efficient cellular delivery and target engagement assessment.
DOI 10.1021/acschembio.5c00702