Systematic identification of engineered methionines and oxaziridines for efficient, stable, and site-specific antibody bioconjugation
S. K. Elledge, H. L. Tran, A. H. Christian, V. Steri, B. Hann, F. D. Toste, C. J. Chang, J. A. Wells
This study systematically identifies engineered methionines and oxaziridines for efficient, stable, and site-specific antibody bioconjugation, finding stable sulfimide modifications comparable to cysteine-maleimide conjugation.
bioRxiv · Aug 28, 2019Bioengineering