Pharmacology & ToxicologybioRxivPreprint
DIFFERENTIAL ACTIVATION OF G-PROTEIN SUBTYPES BY DOPAMINE D1 RECEPTOR ALLOSTERIC MODULATION
Anh Minh Nguyen, Hayato Umaoka, Hideaki Yano
This study investigates how LY3154207, a D1R PAM, differentially activates G-protein subtypes and shows it enhances Gs signaling and selectivity of agonists.
DOI 10.64898/2026.09.26.754724