Gαq-stimulated gene expression is insensitive to Bromo extra terminal domain inhibitors in HEK 293 cells
Ashika Jain, Viviane Pagé, Dominic Devost, Darlaine Pétrin, Terence E. Hébert, Jason C. Tanny
The paper tests BET protein responsiveness to G protein isoforms in HEK 293 cells and finds Gq-induced gene expression is insensitive to BET inhibitors, while Gs-induced expression is sensitive to BET degradation.
International Journal of Molecular Sciences · Sep 12, 2025Peer-reviewedMolecular Biology