Molecular mapping and functional validation of GLP-1R cholesterol binding sites in pancreatic beta cells
Affiong Ika Oqua, Kin Chao, Liliane El Eid, Lisa Casteller, Billy P Baxter, Alba Miguéns‐Gómez, Sebastian Barg, Ben J. Jones, Jorge Bernardino de la Serna, Sarah L. Rouse, Alejandra Tomás
This study identifies and validates cholesterol binding sites on GLP-1R in pancreatic beta cells, showing their role in receptor function and potential for drug design.
eLife · Apr 24, 2025Peer-reviewedCell Biology