Divergent effects of target protein stabilisation versus overproduction on PROTAC activity
Evelina Gudauskaite, Brianda Hernandez Moran, Gillian C.A. Taylor, Andrew J. Wood
This study compares how stabilizing versus overproducing target proteins affects PROTAC activity using β-catenin as a model.
bioRxiv · Apr 18, 2026 · PreprintCancer Biology