LiP-Quant, an automated chemoproteomic approach to identify drug targets in complex proteomes
Ilaria Piazza, Nigel Beaton, Roland Bruderer, Thomas Knobloch, Crystel Barbisan, Isabella Siepe, Oliver Rinner, Natalie de Souza, Paola Picotti, Lukas Reiter
LiP-Quant identifies drug targets in complex proteomes using limited proteolysis and mass spectrometry, providing EC50 estimates and distinguishing between homologous proteins.
bioRxiv · Dec 1, 2019 · PreprintSystems Biology