Pharmacological characterization and radiolabeling ofVUF15485, a high-affinity small-molecule agonist for theatypical chemokine receptor ACKR3
A. Zarca, I. Adlere, C. P. Viciano, M. Arimont-Segura, M. Meyrath, I. A. Simon, J. P. M. Bebelman, D. Laan, H. G. J. Custers, E. C. Janssen, K. L. Versteegh, R. Bosma, I. J. P. De Esch, H. F. Vischer, M. Wijtmans, , R. Leurs
This paper characterizes VUF15485, a high-affinity ACKR3 agonist, and reports its radiolabeling and binding properties.
bioRxiv · Jul 12, 2023Pharmacology & Toxicology