Mechanism of small molecule inhibition of Plasmodium falciparum myosin A informs antimalarial drug design
Dihia Moussaoui, James P. Robblee, Julien Robert‐Paganin, Daniel Auguin, Fabio Fisher, Patricia M. Fagnant, Jill E. Macfarlane, Julia Schaletzky, Eddie Wehri, Christoph Mueller‐Dieckmann, Jake Baum, Kathleen M. Trybus, Anne Houdusse
This paper identifies a small molecule inhibitor of Plasmodium falciparum myosin A, showing it blocks ATP hydrolysis and parasite growth.
Nature Communications · Jun 12, 2023Peer-reviewedMolecular Biology