Identification of first-in-class small molecule potential inhibitor of GDF15
Antonio Chiariello, Lorenzo Lenti, Lorenzo Trofarello, Manuela Sollazzo, Mattia Lauriola, Alberto Del Río, Stefano Salvioli, Marco Daniele Parenti, Maria Conte
This study identifies a small molecule inhibitor of GDF15 through in silico screening and validates its effects on cancer and normal cells.
bioRxiv · Dec 14, 2025 · PreprintMolecular Biology