1,2,4-Triazole-based first-in-class non-nucleoside inhibitors of bacterial enzyme MraY
Tomayo I. Berida, Tzu‐Yu Huang, Stefanie C. Weck, Marcel Lutz, Samuel R. McKee, Nathalie Kagerah, Destinee L. Manning, Mohamed E. Jahan, Sushil K. Mishra, Jennifer E. Herrmann, Rolf Müller, Robert J. Doerksen, Christina L. Stallings, Christian Ducho, Sudeshna Roy
This paper discovers first-in-class 1,2,4-triazole-based non-nucleoside inhibitors of MraY with broad-spectrum antibacterial activity against multiple bacterial species.
ACS Bio & Med Chem Au · Sep 19, 2025Peer-reviewedBiochemistry