BiochemistrybioRxivPreprint
Molecular Dynamics-Guided Design and Chemoproteomic Profiling of Covalent Kinase Activity Probes
Pratyasha Chakraborty, Anthony J. Carlos, Trayder Thomas…·Raymond E. Moellering
This paper designs and tests covalent kinase activity probes using computational methods and shows they target multiple kinases in live cells with distinct kinetics and conformations.
DOI 10.1101/2025.10.17.683178