Overcoming insecticide resistance through computational inhibitor design
G. Correy, D. Zaidman, A. Harmelin, S. Carvalho, P. D. Mabbitt, V. Calaora, P. J. James, A. C. Kotze, N. London, C. J. Jackson
The paper designs boronic acid inhibitors to overcome insecticide resistance by targeting carboxylesterases in pests, significantly enhancing insecticide efficacy and reducing usage.
bioRxiv · Jan 24, 2019Biochemistry