BiophysicsbioRxiv
Allosteric modulation of the adenosine A2A receptor by cholesterol
S. K. Huang, O. Almurad, R. J. Pejana…·R. S. Prosser
This study shows cholesterol weakly modulates A2AR conformation and signaling through indirect membrane effects rather than direct allosteric binding.
DOI 10.7554/elife.73901