TRPV1 regulates opioid analgesia during inflammation
Lilian Basso, Reem Aboushousha, Churmy Y. Fan, Mircea Iftinca, Helvira Melo, Robyn E. Flynn, Francina Agosti, Morley Donald Hollenberg, Roger J. Thompson, Emmanuel Bourinet, Tuan Trang, Christophe Altier
The paper shows TRPV1 channels enhance opioid analgesia during inflammation by promoting beta-arrestin2 nuclear translocation, preventing receptor desensitization.
bioRxiv · Mar 1, 2018 · PreprintNeuroscience