Helical foldamers as selective G-quadruplex ligands
Alexander König, Vincent Laffilé, Stéphane Thore, Cameron D. Mackereth, Liliya A. Yatsunyk, Yann Ferrand, Eric Largy, Valérie Gabelica
This study identifies helical foldamers with quinoline and pyridine units as selective G-quadruplex ligands, showing preference for parallel structures and sequence variants.
bioRxiv · Feb 25, 2025 · PreprintBiophysics