Engineering Stapled Peptide Inhibitors Reveals Design Principles for Targeting Talin-Induced Integrin Activation
Tong Gao, Elizaveta Belova, Yujiro MORI, Kathrine Wang, William H. Deni, Heinrich Röder, Bojana Gligorijevic, Jinhua Wu
The paper designs stapled peptides targeting talin-induced integrin activation, showing improved binding and cell uptake in optimized versions.
bioRxiv · Aug 31, 2026 · PreprintBiochemistry