C-6 Modified 2-F-Fucose Derivatives as Inhibitors of Fucosyl Transferases
The paper designs and evaluates C-6 modified GDP-2-F-Fuc analogs as FUT inhibitors, finding two compounds that potently inhibit FUT1, 3, 6, and 9 with minimal activity against FUT8.
ChemBioChem · Oct 13, 2025Peer-reviewedBiochemistry