Impact of GPR39 Inhibition on Tissue Oxygen Tension in Acute Myocardial Infarction: Modeling Using an Indirect Response Pharmacokinetics/Pharmacodynamics Approach
Davide Ronchi, Chiara Roversi, Simone Zannoni…·Sanjiv Kaul
This paper develops a population PK/PD model to simulate the effects of VC108, a GPR39 inhibitor, on myocardial oxygen tension during acute myocardial infarction and reperfusion.