IGF2 Peptide-Based LYTACs for Targeted Degradation of Extracellular and Transmembrane Proteins
Michał Mikitiuk, Jan Barczyński, Przemysław Bielski, Marcelino Arciniega, Urszula Tyrcha, Aleksandra Hec, Andrea D. Lipińska, Michał Rychłowski, Tad A. Holak, Tomasz Sitar
This paper develops IGF2-based LYTACs for lysosomal degradation of extracellular and transmembrane proteins, showing enhanced in vitro effects compared to anti-PD-L1 antibodies.
Molecules · Nov 10, 2023Peer-reviewedMolecular Biology