Cancer BiologybioRxivPreprint
Development and characterization of Novel Small Molecule Inhibitors Targeting LAG-3 Protein
Oleksandr Yakovenko, Alireza Baradaran‐Heravi, Steven J.M. Jones
This paper develops and characterizes small-molecule inhibitors of LAG-3, a protein that suppresses antitumor immunity, using a novel semi-allosteric mechanism.
DOI 10.1101/2025.08.29.673196