BiochemistryJACS AuPeer-reviewed
Influence of Macrocyclization Strategies on DNA-Encoded Cyclic Peptide Libraries
Hanqing Zhao, Xue Li, Xueyu Yao…·Xiaojie Lu
This study evaluates how different macrocyclization strategies affect DNA-encoded cyclic peptide library selections against MDM2 and GIT1, identifying potent inhibitors and elucidating binding mechanisms.
13 citations