Cancer BiologybioRxivPreprint
AI-Driven Computational Design of Peptide-Based WWP1 Inhibitors as Promising Therapeutic Agents Against Breast Cancer, Including Triple-Negative Subtype
Enrico Mario Alessandro Fassi, Sara Mathlouthi, Elena Maspero…·Giovanni Grazioso
This study uses AI to design a peptide inhibitor of WWP1, showing potent activity against breast cancer, especially TNBC, with promising cytotoxic effects and synergistic potential with PI3K inhibitors.
DOI 10.64898/2026.08.08.742959