Diverse Ligands for Mycobacterial CYP124 Identified from Plant and Marine Compounds
Leonid A. Kaluzhskiy, Evgeniy O. Yablokov, Tatsiana Varaksa, Anna V. Grudo, A. I. Karputs, Irina P. Grabovec, Yuri V. Mezentsev, Elena Zelepuga, Oksana V. Gnedenko, Dmitriy K. Tolkanov, Timofey V. Malyarenko, Sophia A. Kolesnikova, Anastasia B. Kozhushnaya, Е. А. Васильева, Natalia Mishchenko, , Alexis Ivanov
The paper identifies nine novel non-azole ligands for Mycobacterium tuberculosis CYP124 from plant and marine compounds, revealing potential for mechanism-based tuberculosis inhibitors.
Biochimie · Feb 26, 2026Peer-reviewedBiochemistry