The mycotoxin Beauvericin is an uncompetitive inhibitor of Cathepsin B
Xiaoli Yang, Pablo Cea‐Medina, Mohanraj Gopalswamy, Aparna Vaidya, Sonja Schavier, Shixin Oltzen, Sofie Moßner, Anfei Huang, Jing Qi, Johanna Maria Hölken, Nicole Elisabeth Teusch, Doreen Manuela Floss, Markus Uhrberg, Holger Gohlke, Stefanie Scheu
This study identifies Beauvericin as an uncompetitive inhibitor of Cathepsin B through NMR, enzyme kinetics, and molecular docking analyses in dendritic cells.
Protein Science · May 24, 2025Peer-reviewedBiochemistry