Selective Peptidomimetic Inhibitors of NTMT1/2: Rational design, synthesis, characterization, and crystallographic studies
B. D. Mackie, D. Chen, G. Dong, C. Dong, H. Parker, N. Noinaj, C. E. Schaner Tooley, J. Min, R. Huang
This paper designs and characterizes peptidomimetic inhibitors of NTMT1/2, showing high selectivity and cell-permeable activity.
bioRxiv · Apr 13, 2020Biochemistry