Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX
A. Vaskevicius, D. Baronas, J. Leitans, A. Kvietkauskaite, A. Ruksenaite, E. Manakova, Z. Toleikis, A. Kaupinis, A. Kazaks, M. Gedgaudas, A. Mickeviciute, V. Juozapaitiene, H. Schioth, K. Jaudzems, M. Valius, , D. Matulis
The paper designs and tests novel covalent inhibitors targeting CAIX, achieving high affinity and selectivity for cancer treatment.
bioRxiv · May 20, 2024Biophysics